5-HT Receptor


5-HT receptors (5-hydroxytryptamine receptors,The serotonin receptors) are a group of G protein-coupled receptors (GPCRs) and ligand-gated ion channels (LGICs) found in the central and peripheral nervous systems. They mediate both excitatory and inhibitory neurotransmission. The serotonin receptors are activated by the neurotransmitter serotonin, which acts as their natural ligand.

  • Donitriptan hydrochloride EI1027

    Donitriptan hydrochloride是5-HT1B/1D 激动剂。

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  • Dolasetron mesylate EI1022

    Dolasetron mesylate是活性选择性 5-HT3 拮抗剂。

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  • DOI hydrochloride EI1021

    DOI hydrochloride是Mixed 5-HT2A/2C 激动剂。

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  • DOB hydrochloride EI1018

    DOB hydrochloride是选择性 5-HT2 激动剂。

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  • Dexfenfluramine hydrochloride EI0962

    Dexfenfluramine hydrochloride是5-HT uptake inhibitor(摄取抑制剂),也能促进5-HT 的释放。

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  • Donitriptan hydrochloride EI1027

    Donitriptan hydrochloride是5-HT1B/1D 激动剂。

    More
  • Dolasetron mesylate EI1022

    Dolasetron mesylate是活性选择性 5-HT3 拮抗剂。

    More
  • DOI hydrochloride EI1021

    DOI hydrochloride是Mixed 5-HT2A/2C 激动剂。

    More
  • DOB hydrochloride EI1018

    DOB hydrochloride是选择性 5-HT2 激动剂。

    More
  • Dexfenfluramine hydrochloride EI0962

    Dexfenfluramine hydrochloride是5-HT uptake inhibitor(摄取抑制剂),也能促进5-HT 的释放。

    More
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